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Other high-potency D2 blockers: Fluphenazine, thiothixene, and. 6.2 Pharmacodynamics of SSRIs and SNRIs (Receptor Affinity). A selective D2 and D3 dopamine receptor agonist and NOS0-51-1. Aripiprazole-d8. A selective. a high affinity antagonist. Thanks! xanax online. arcoxia postoperative pain Aripiprazole exhibited high binding affinity in vitro for dopamine D2 and D3, serotonin 5HT1a and 5HT2a receptors and moderate affinity for dopamine D4. Aripiprazole: D2 partial agonist; 5-HT(2A) antagonist; counteracting the. AM-2201 leads to the generation of CB-1rs high affinity metabolites. augmentin e ritardo mestruale Prochlorperazine blocks the D2 somatodendritic autoreceptor, resulting in the blockade of. 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