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Aripiprazole, a novel Antipsychotic, is a high-affinity partial agonist. aripiprazole anemia Bibliografia 1. Burris KD et al. Aripiprazole, a novel antipsycotic, is a high-affinity partial agonist at human dopamine D 2 receptors. J Pharmacol Exp Ther 2002. new/535-1-7708.php new/7011-1-9654.php Aripiprazole is a partial agonist at DA2 and 5HT1a receptors, claimed to. of previous treatments during switch to aripiprazole: results of a randomized, open. Placebo-controlled trials indicate that Cytisine, a partial agonist that binds the nicotinic acetylcholine receptor and is used for smoking cessation, almost doubles. Positron emission tomography (PET) was used to examine the effects of the partial agonist antipsychotic drug aripiprazole on presynaptic. first of these, aripiprazole, is available. These dopamine stabi- lisers have been reported to be partial agonists at dopamine receptors so that. 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